doc. RNDr. Miroslav SOURAL, Ph.D.

Zástupný obrázek
Kontaktní údaje

585634405

Katedra organické chemie

Přírodovědecká fakulta

17. listopadu 12

3.015

docent

ČLÁNEK
Ondrová K., Zůvalová I., Vyhlídalová B., Krasulová K., Miková E., Vrzal R., Nádvorník P., Kopečná M., Kopečný D., Šebela M., Soural M., Dvořák Z. Monoterpenoid aryl hydrocarbon receptor allosteric antagonists protect against ultraviolet skin damage in female mice. Nature Communications. 2023.
Sládeková L., Zgarbová E., Vrzal R., Vanda D., Soural M., Dvořák Z. Switching on/off aryl hydrocarbon receptor and pregnane X receptor activities by chemically modified tryptamines. TOXICOLOGY LETTERS. 2023.
Lemrová B., Maloň M., Soural M. Efficient Synthesis of Pentasubstituted Pyrroles via intramolecular C-arylation. Organic and Biomolecular Chemistry. 2022.
Řezníčková E., Krajčovičová S., Peřina M., Kovalová M., Soural M., Kryštof V. Modulation of FLT3-ITD and CDK9 in acute myeloid leukaemia cells by novel proteolysis targeting chimera (PROTAC). EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 2022.
Králová P., Žáková K., Pospíšilová L., Soural M. Synthesis of 2,3-Disubstituted Quinoline-4-carbonitriles through Truce–Smiles Rearrangement of Phenacyl-4-nitrobenzenesulfonamides. European Journal of Organic Chemistry (online). 2022.
Kriegelsteinová P., Lemrová B., Ručilová V., Soural M. Copper-free solid-phase synthesis of triazolo[1,5-a][1,4]diazepin-6-ones. Advanced Synthesis & Catalysis. 2021.
Maková B., Mik V., Lišková B., Gonzalez G., Vítek D., Medvedíková M., Ručilová V., Kadlecová A., Gándara Barreiro Z., Zatloukal M., Soural M., Paruch K., Hajdúch M., Strnad M., Voller J. Cytoprotective activities of kinetin purine isosteres. Bioorganic and Medicinal Chemistry. 2021.
Ručilová V., Šwierczek A., Vanda D., Funk P., Lemrová B., Soural M. New Imidazopyridines with Phosphodiesterase 4 and 7 Inhibitory Activity and Their Efficacy in Animal Models of Inflammatory and Autoimmune Diseases. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 2021.
Krajčovičová S., Jorda R., Vanda D., Soural M., Kryštof V. 1,4,6-Trisubstituted imidazo[4,5-c]pyridines as inhibitors of Bruton’s tyrosine kinase. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 2021.
Krajčovičová S., Danišková A., Bendová K., Nový Z., Soural M., Petřík M. [68Ga]Ga-DFO-c(RGDyK): synthesis and evaluation of its potential for tumor imaging in mice. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES. 2021.
Králová V., Soural M., Horák R., Hradil P. Convenient Synthesis of Furo[3,2-b]quinolin-4(1H)-ones. SYNLETT. 2020.
Králová P., Maloň M., Pospíšil J., Soural M. Rearrangement of Threonine and Serine-Based N-(3-Phenylprop-2-yn-1-yl) Sulfonamides Yields Chiral Pyrrolidin-3-ones. JOURNAL OF ORGANIC CHEMISTRY. 2020.
Jorda R., Krajčovičová S., Králová P., Soural M., Kryštof V. Scaffold hopping of the SYK inhibitor entospletinib leads to broader targeting of the BCR signalosome. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 2020.
Horák R., Kořistek K., Šamšulová V., Slaninová L., Grepl M., Kvapil L., Funk P., Hradil P., Soural M. Structural analogues of quinoline alkaloids: Straightforward route to [1,3]dioxolo[4,5-c]quinolines with antibacterial properties. Journal of Heterocyclic Chemistry. 2020.
Králová P., Lemrová B., Maloň M., Soural M. Synthesis of Chiral 1,4-Oxazepane-5-Carboxylic Acids from Polymer-Supported Homoserine. RSC Advances. 2020.
Frömmel J., Končitíková R., Kopečný D., Soural M., Šebela M. Oxidation of imidazole- and pyrazole-derived aldehydes by plant aldehyde dehydrogenases from the family 2 and 10. CHEMICO-BIOLOGICAL INTERACTIONS. 2019.
Králová P., Benická S., Soural M. Polymer-assisted Synthesis of Single and Fused Diketomorpholines. ACS Combinatorial Science. 2019.
Krajčovičová S., Jorda R., Hendrychová D., Kryštof V., Soural M. Solid-phase synthesis for thalidomide-based proteolysis-targeting chimeras (PROTAC). CHEMICAL COMMUNICATIONS. 2019.
Bürglová K., Rylová G., Markos A., Přichystalová H., Soural M., Petráček M., Medvedíková M., Tejral G., Sopko B., Hradil P., Džubák P., Hajdúch M., Hlaváč J. Identification of Eukaryotic Translation Elongation Factor 1-alpha 1 Gamendazole-Binding Site for Binding of 3-Hydroxy-4(1. JOURNAL OF MEDICINAL CHEMISTRY. 2018.
Vanda D., Soural M., Canale V., Chaumont-Dubel S., Satala G., Kos T., Funk P., Fülöpová V., Lemrová B., Koczurkiewicz P., Pekala E., Bojarski AJ., Popik P., Marin P., Zajdel P. Novel non-sulfonamide 5-HT6 receptor partial inverse agonist in a group of imidazo[4,5-b]pyridines with cognition enhancing properties. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 2018.
Králová P., Ručilová V., Soural M. Polymer-Supported Syntheses of Heterocycles Bearing Oxazine and Thiazine Scaffolds. ACS Combinatorial Science. 2018.
Ručilová V., Soural M. Recent advances in the applications of triethylsilane in organic synthesis. SYNTHESIS-STUTTGART. 2018.
Horák R., Kvapil L., Motyka K., Slaninová L., Grepl M., Kořistek K., Urbášek M., Hradil P., Soural M. Synthesis of 2-alkenyl-3-hydroxyquinolin-4(1H)-ones as promising antimicrobial and fluorescent agents. TETRAHEDRON. 2018.
Krajčovičová S., Stanková J., Džubák P., Hajdúch M., Soural M., Urban M. Synthetic approach for rapid preparation of BODIPY conjugates and their use in imaging of cellular drug uptake and distribution. CHEMISTRY-A EUROPEAN JOURNAL. 2018.
Krajčovičová S., Gucký T., Hendrychová D., Kryštof V., Soural M. A Stepwise Approach for the Synthesis of Folic Acid Conjugates with Protein Kinases Inhibitors. Journal of Organic Chemistry. 2017.
Králová P., Maloň M., Volná T., Ručilová V., Soural M. Polymer-supported Stereoselective Synthesis of Benzoxazino[4,3-b][1,2,5]thiadiazepinone-6,6-dioxides. ACS Combinatorial Science. 2017.
Králová P., Fülöpová V., Maloň M., Volná T., Popa I., Soural M. Stereoselective polymer-supported synthesis of morpholine and thiomorpholine-3-carboxylic acid derivatives. ACS Combinatorial Science. 2017.
Funk P., Motyka K., Soural M., Maloň M., Koshino H., Joachim K., Hlaváč J. Study of 2-aminoquinolin-4(1H)-one under Mannich and Retro-Mannich Reaction. PLoS One. 2017.
Ručilová V., Králová P., Soural M. Synthesis of Disubstituted Pyrazino-Oxazine Derivatives with Controlled Stereochemistry. European Journal of Organic Chemistry (online). 2017.
Fülöpová V., Soural M. Solid-phase synthesis of heterocycles with the use of α--haloketones as the key building blocks. Synthesis: journal of synthetic organic chemistry. 2016.
Krajčovičová S., Soural M. Solid-phase synthetic strategies for the preparation of purine derivatives. ACS Combinatorial Science. 2016.
Rylová G., Oždian T., Varanasi L., Soural M., Hlaváč J., Holub D., Džubák P., Hajdúch M. Affinity-Based Methods in Drug-Target Discovery. Current Drug Targets. 2015.
Soural M., Hodoň J., Dickinson N., Šidová V., Gurská S., Džubák P., Hajdúch M., Šarek J., Urban M. Preparation of conjugates of cytotoxic lupane triterpenes with biotin. Bioconjugate Chemistry. 2015.
Funk P., Motyka K., Džubák P., Znojek P., Gurská S., Kusz J., Mcmaster C., Hajdúch M., Soural M. Preparation of 2-Phenyl-3-hydroxyquinoline-4(1H)-one-5-carboxamides as Potential Anticancer and Fluorescence Agents. RSC Advances (online). 2015.
Buzgo M., Greplová J., Soural M., Bezděková D., Míčková A., Kofroňová O., Benada O., Hlaváč J., Amler E. PVA immunonanofibers with controlled decay. Polymer. 2015.
Vanda D., Jorda R., Lemrová B., Volná T., Kryštof V., Mcmaster C., Soural M. Synthesis of Novel N-9-Substituted Purine Derivatives from Polymer Supported alpha-Amino Acids. ACS Combinatorial Science. 2015.
Vanda D., Jorda R., Lemrová B., Volná T., Kryštof V., Mcmaster C., Soural M. Synthesis of novel N9-substituted purine derivatives from polymer supported α-amino acids. ACS Combinatorial Science. 2015.
Lemrová B., Soural M. Synthetic strategies for preparing bicyclic guanidines. European Journal of Organic Chemistry. 2015.
Lemrová B., Smyslová P., Popa I., Oždian T., Zajdel P., Soural M. Directed Solid-Phase Synthesis of Trisubstituted Imidazopyridines and Imidazopyridines. ACS Combinatorial Science. 2014.
Hartmanová L., Fryčák P., Soural M., Tureček F., Havlíček V., Lemr K. Ion internal energy, salt tolerance and a new technical improvement of desorption nanoelectrospray. Journal of Mass Spectrometry. 2014.
Mcmaster C., Fülöpová V., Popa I., Grepl M., Soural M. Solid-Phase Synthesis of Anagrelide Sulfonyl Analogues. ACS Combinatorial Science. 2014.
Messina I., Popa I., Maier V., Soural M. Solid-Phase Synthesis of 5-Noranagrelide Derivatives. ACS Combinatorial Science. 2014.
Kadrič J., Motyka K., Džubák P., Hajdúch M., Soural M. Synthesis, cytotoxic activity and fluorescence properties of a set of novel 3-hydroxyquinolin-4(1H)-ones. Tetrahedron Letters. 2014.
Kopečný D., Končitíková R., Tylichová M., Vigouroux A., Moskalíková H., Soural M., Šebela M., Moréra S. Plant ALDH10 family: identifying critical residues for substrate specificity and trapping a thiohemiacetal intermediate. Journal of Biological Chemistry. 2013.
Soural M., Hradil P., Křupková S., Hlaváč J. An Interesting Synthetic Pathway to Some Quinolin-4(1H)ones: Phenacylanthranilates Rearrangement – Limits and Scopes. Mini - Reviews in Organic Chemistry. 2012.
Frömmel J., Soural M., Tylichová M., Kopečný D., Demo G., Wimmerová M., Šebela M. Plant aminoaldehyde dehydrogenases oxidize a wide range of nitrogenous heterocyclic aldehydes. Amino Acids. 2012.
Fülöpová V., Gucký T., Grepl M., Soural M. Solid-Phase Synthesis of Trisubstituted Benzo[1,4]-Diazepin-5-one Derivatives. ACS Combinatorial Science. 2012.
ONDRA P., SOKOLOVÁ B., STAŇKOVÁ M., SOURAL M., HEBKÁ L., LEMR K., STŘÍBRNÝ J. Determination of muscarine in human urine by electrospray liquid chromatographic-mass spectrometric. Journal of Chromatography. B, Analytical Technologies in the Biomedical and Life Sciences. 2011.
VAŇKOVÁ B., KRCHŇÁK V., SOURAL M., HLAVÁČ J. Direct C-H Arylation of Purine on Solid Phase and Its Use for Chemical Libraries Synthesis. ACS Combinatorial Science. 2011.
MOTYKA K., HLAVÁČ J., SOURAL M., HRADIL P., Krejčí P., Kvapil L., Weiss M. Fluorescence properties of some 2-(4-aminosubstituted-3-nitrophenyl)-3-hydroxyquinolin-4(1H)-ones. Tetrahedron Letters. 2011.
CANKAŘOVÁ N., FUNK P., HLAVÁČ J., SOURAL M. Novel preloaded resins for solid-phase biotinylation of carboxylic acids. Tetrahedron Letters. 2011.
MOTYKA K., VAŇKOVÁ B., HLAVÁČ J., SOURAL M., FUNK P. Purine Scaffold Effect on Fluorescence Properties of Purine-Hydroxyquinolinone Bisheterocycles. Journal of Fluorescence. 2011.
SOURAL M., HLAVÁČ J., FUNK P., DŽUBÁK P., HAJDÚCH M. 2-Phenylsubstituted-3-Hydroxyquinolin-4(1H)-one-Carboxamides: Structure-Cytotoxic Activity Relationship Study. ACS Combinatorial Science. 2011.
Motyka K., Hlaváč J., Soural M., Funk P. Fluorescence properties of 2-aryl-3-hydroxyquinolin-4(1H)-one-carboxamides. Tetrahedron Letters. 2010.
Vičar J., Soural M., Hlaváč J. SEPARACE KVARTÉRNÍCH BENZO[c]FENANTHRIDINOVÝCH ALKALOIDŮ Z Macleaya cordata. Chemické listy. 2010.
Vaňková B., Hlaváč J., Soural M. Solid-phase Synthesis of Highly Diverse Purine-Hydroxyquinolinone Bisheterocycles. Journal of Combinatorial Chemistry. 2010.
Soural M., Funk P., Kvapil L., Hradil P., Hlaváč J., Bertolasi V. Study of anthranilate cyclisation to 2-hydroxymethyl-2,3-dihydro-quinazolin-4(1H)-ones and an alternative synthetic route. Arkivoc. 2010.
Soural M., Hlaváč J., Hradil P., Hajdúch M. Efficient Synthesis and Cytotoxic Activity of Some Symmetrical Disulfides Derived from the Quinolin-4(1H)-one Skeleton. European Journal of Organic Chemistry. 2009.
Soural M., Hlaváč J., Hradil P., Hajdúch M. Efficient Synthesis and Cytotoxic Activity of Some Symmetrical Disulfides Derived from the Quinolin-4(1H)-one Skeleton. European Journal of Organic Chemistry (online). 2009.
Soural M., Hlaváč J., Hradil P., Hajdúch M. Efficient Synthesis and Cytotoxic Activity of Some Symmetrical Disulfides Derived from the Quinolin-4(1H)-one Skeleton. European Journal of Organic Chemistry (online). 2009.
Bouillon I., Soural M., Miller M.J.., Krchňák V. Resins with Identical Specifications Are Not Identical. Identifying a Useful Solid-Phase Resin. Journal of Combinatorial Chemistry. 2009.
Křupková S., Soural M., Hlaváč J., Hradil P. Solid-Phase Synthesis of 3-Hydroxy-6-Nitroquinolin-4(1H)-ones with Two Diversity Positions. Journal of Combinatorial Chemistry. 2009.
Hradil P., Hlaváč J., Soural M., Hajdúch M., Kolář M., Večeřová R. 3-Hydroxy-2-phenyl-4(1H)-quinolinones as promising biologically active compounds. Mini - Reviews in Medicinal Chemistry. 2009.
Hradil P., Hlaváč J., Soural M., Hajdúch M., Kolář M., Večeřová R. 3-Hydroxy-2-phenyl-4(1H)-quinolinones as promising biologically active compounds. Mini - Reviews in Medicinal Chemistry. 2009.
Soural M., Bouillon I., Krchňák V. Combinatorial Libraries of Bis-heterocyclic Compounds with Skeletal Diversity. Journal of Combinatorial Chemistry. 2008.
Bouillon I., Soural M., Krchňák V. Resin Capsules: Permeable Containers for Parallel/Combinatorial Solid-Phase Organic Synthesis. Journal of Combinatorial Chemistry. 2008.
Stýskala J., Cankař P., Soural M., Bednář P., Lemr K. Synthesis of some deuterated dialkylaminoethyls as possible standards for the mass spectrometric monitoring of chemical warfare agents. Journal of Labelled Compounds and Radiopharmaceuticals. 2008.
Stýskala J., Cankař P., Soural M., Bednář P., Lemr K. Preparation and characterization of some unsymmetrical 2-(dialkylamino)ethanethiols. Arkivoc. 2007.
Stýskala J., Cankař P., Soural M., Hlaváč J., Hradil P., Vičar J., Šimánek V. Synthesis of isodecarine. Heterocycles. 2007.
Stýskala J., Cankař P., Soural M., Hlaváč J., Hradil P., Vičar J., Šimánek V. Synthesis of isodecarine. Heterocycles. 2007.
Hradil P., Grepl M., Hlaváč J., Soural M., Maloň M., Bertolasi V. Some new routes for the preparation of 3-amino-2-phenyl-4(1H)-quinolinones from anthranilamides. Journal of Organic Chemistry. 2006.
Soural M., Hlaváč J., Hradil P., Fryšová I., Hajdúch M., Bertolasi V., Maloň M. Synthesis and cytotoxic activity of substituted 2-phenyl-3-hydroxy-4(1H)-quinolinones-7-carboxylic acids and their phenacyl esters. European Journal of Medicinal Chemistry. 2006.
Soural M., Hlaváč J., Hradil P., Fryšová I., Hajdúch M., Bertolasi V., Maloň M. Synthesis and cytotoxic activity of substituted 2-phenyl-3-hydroxy-4(1H)-quinolinones-7-carboxylic acids and their phenacyl esters. European Journal of Medicinal Chemistry. 2006.
Spáčilová L., Hlaváč J., Hradil P., Fryšová I., Maloň M., Soural M., Krejčí P. Synthesis of N-amino-3-hydroxy-2-phenyl-4(1H)-quinolinone. Journal of Heterocyclic Chemistry. 2006.
Soural M., Hlaváč J., Hradil P., Hajdúch M. Syntéza a cytotoxické účinky vícejaderných derivátů 3-hydroxy-4(1H)-chinolonů. ChemZi. 2005.
PŘÍSPĚVEK VE SBORNÍKU
Hradil P., Hlaváč J., Krejčí P., Soural M., Krchňák V., Hajdúch M., Okawara T. Anticancer activity of 2-substituted 3-hydroxy-4(1H)-quinolinones. Frontiers in CNS and Oncology Medicinal Chemistry. 2007.
Soural M., Hlaváč J., Hradil P., Hajdúch M., Bertolasi V. Synthesis of Substituted 2-Phenyl-3-Hydroxy-4(1H)-Quinolinones Substituted with Carboxylic Group and Their Cytotoxicity Screening. 20th International Congress of Heterocyclic Chemistry. 2005.
KAPITOLA V KNIZE
Fülöpová V., Soural M. Solid-Phase Synthesis of Seven-Membered Heterocycles with Two Nitrogen Atoms. In Krchňák V. (Eds.) Solid-Phase Synthesis of Nitrogenous Heterocycles. Topics in Heterocyclic Chemistry. 2017.
Hlaváč J., Soural M., Krchňák V. Practical Aspects of Combinatorial Solid-Phase Synthesis. Solid-Phase Organic Synthesis: Concepts, Strategies and Applications. 2012.
Soural M., Hlaváč J., Krchňák V. Linkers for Solid-Phase Peptide Synthesis. In Hughes AB. (Eds.) Amino Acids, Peptides and Proteins in Organic Chemistry: Volume 3 - Building Blocks, Catalysis and Coupling Chemistry. 2010.
ABSTRAKT
Řehulka J., Urban M., Krajčovičová S., Soural M., Džubák P., Hajdúch M. Applications of betulinic acid conjugates in drug target research. IMTM REACTOR ABSTRACT BOOK 2019. 2019.
Řehulka J., Urban M., Krajčovičová S., Soural M., Džubák P., Hajdúch M. Applications of betulinic acid conjugates to explore its mode of action. XV. DIAGNOSTIC, PREDICTIVE AND EXPERIMENTAL ONCOLOGY DAYS: ABSTRACT BOOK. 2019.
Urban M., Hodoň J., Borková L., Pokorný J., Krajčovičová S., Lišková B., Soural M., Václavková J., Stanková J., Holub D., Džubák P., Hajdúch M., Šarek J., Řehulka J. Cytotoxic triterpenes and triterpenic conjugates used for studies of mechanisms of action. ABSTRACT BOOK XIV. DIAGNOSTIC, PREDICTIVE AND EXPERIMENTAL ONCOLOGY DAYS. 2018.
Řehulka J., Urban M., Soural M., Hajdúch M., Džubák P. Identifying cellular targets of betulinic acid conjugates. ABSTRACT BOOK XIV. DIAGNOSTIC, PREDICTIVE AND EXPERIMENTAL ONCOLOGY DAYS. 2018.
Urban M., Borková L., Pokorný J., Džubák P., Hajdúch M., Soural M., Šarek J., Krajčovičová S., Řehulka J., Hodoň J. Semisynthetic triterpenic heterocycles with antitumor properties and their mechanism of action. 17th Blue Danube Symposium on Heterocyclic Chemistry. 2017.
Urban M., Hodoň J., Soural M., Václavková J., Holub D., Džubák P., Šarek J., Řehulka J., Hajdúch M. Semisynthetic triterpenoid heterocycles - synthesis, cytotoxicity, and studies of their mechanism of action. Abstract Book: XIII. Diagnostic, Predictive and Experimental Oncology Days. 2017.
Polishchuk P., Džubák P., Konečný P., Frydrych I., Doležal D., Purová D., Soural M., Hlaváč J., Rylová G., Hajdúch M. Activity profile analysis of carboxamides of 2-aryl-3-hdyroxyquinolin-4(1H)-one. XI. Diagnostic, Predictive and Experimental Oncology Days: Abstract Book. 2015.
Rylová G., Džubák P., Janošťáková A., Frydrych I., Konečný P., Holub D., Oždian T., Doležal D., Soural M., Hlaváč J., Hajdúch M. Molecular target identification of quinolinone based anticancer compounds. Proceedings of the 105th Annual Meeting of the American Association for Cancer Research. 2014.
Rylová G., Džubák P., Janošťáková A., Frydrych I., Holub D., Oždian T., Doležal D., Soural M., Hlaváč J., Hajdúch M. Biological actitivty and molecular target of quinolinone derivatives with anticancer effect. IX. Diagnostic, Predictive and Experimetnal Oncology Days: Abstract Book. 2013.
Rylová G., Džubák P., Janošťáková A., Frydrych I., Konečný P., Holub D., Oždian T., Doležal D., Soural M., Hlaváč J., Hajdúch M. Biological activity and molecular targets of quinolinone derivatives with anticancer effect. Sborník abstrakt: Konference Chemické biologie a genetiky. 2013.
Rylová G., Džubák P., Janošťáková A., Frydrych I., Konečný P., Holub D., Oždian T., Doležal D., Soural M., Hlaváč J., Hajdúch M. Biological target and molecular activity of quinolinone derivatives with anticancer effect. Chemistry towards Biology: 6th Central Europe Conference. 2013.
Rylová G., Džubák P., Janošťáková A., Frydrych I., Konečný P., Holub D., Oždian T., Doležal D., Soural M., Hlaváč J., Hajdúch M. Biological Activity and Molecular Targets of Quinolinone Derivatives with Anticancer Effect. 6th Central and Eastern European Proteomics Conference: Book of Abstracts and Program. 2012.
Rylová G., Džubák P., Janošťáková A., Frydrych I., Konečný P., Holub D., Oždian T., Doležal D., Soural M., Hlaváč J., Hajdúch M. Identifikace cílů protinádorových léčiv pomocí afinitní purifikace. Optics Communications. 2012.
Rylová G., Džubák P., Janošťáková A., Frydrych I., Konečný P., Holub D., Oždian T., Doležal D., Soural M., Hlaváč J., Hajdúch M. Molecular targets of quinolinone derivatives with anticancer activity. Proceedings: AACR Annual Meeting. 2012.
Rylová G., Džubák P., Janošťáková A., Frydrych I., Konečný P., Holub D., Oždian T., Doležal D., Soural M., Hlaváč J., Hajdúch M. Proteomické metody k identifikaci protinádorových cílů. Sborník přednášek a posterů, program. 2012.
Řehulka J., Džubák P., Frydrych I., Krejčí P., Soural M., Hajdúch M. The role of selected miRNA in MDR caused by P-gp, MRP1 and LRP/MVP in NSCLC patients. Biomedical Papers-Olomouc. 2012.
RYLOVÁ G., DŽUBÁK P., ŠPENEROVÁ M., JANOŠŤÁKOVÁ A., FRYDRYCH I., KONEČNÝ P., HOLUB D., OŽDIAN T., DOLEŽAL D., SOURAL M., HLAVÁČ J., HAJDÚCH M. Biological activity and molecular targets of quinoline derivatives with anticancer effect. Conference book: The Student Scientific Conference on Cancer Research. 2011.
RYLOVÁ G., DŽUBÁK P., ŠPENEROVÁ M., JANOŠŤÁKOVÁ A., FRYDRYCH I., KONEČNÝ P., HOLUB D., OŽDIAN T., DOLEŽAL D., SOURAL M., HLAVÁČ J., HAJDÚCH M. Biological Activity and Molecular Targets of Quinoline Derivatives with Anticancer Effect. Sborník abstrakt konference: Nová léčiva závažných lidských onemocnění. 2011.
RYLOVÁ G., DŽUBÁK P., ŠPENEROVÁ M., JANOŠŤÁKOVÁ A., FRYDRYCH I., KONEČNÝ P., HOLUB D., OŽDIAN T., DOLEŽAL D., SOURAL M., HLAVÁČ J., HAJDÚCH M. Biological activity and protein targets of quinoline derivatives with anticancer effect. Book of Abstracts - 5th Central and Eastern European Proteomic Conference. 2011.
RYLOVÁ G., DŽUBÁK P., ŠPENEROVÁ M., JANOŠŤÁKOVÁ A., FRYDRYCH I., KONEČNÝ P., HOLUB D., OŽDIAN T., DOLEŽAL D., SOURAL M., HLAVÁČ J., HAJDÚCH M. BIOLOGICKÁ AKTIVITA A MOLEKULÁRNÍ CÍLE CHINOLONOVÝCH DERIVÁTŮ S PROTINÁDOROVÝMI ÚČINKY. Chemické listy. 2011.
KONEČNÝ P., DŽUBÁK P., SOURAL M., FRYDRYCH I., RYLOVÁ G., HAJDÚCH M. Flow cytometric profiling of 2-Phenylsubstituted-3-Hydroxyquinolin-4(1H)-one-Carboxamides and their anticancer activities. Towards toxicity assessment without animals. 2011.
RYLOVÁ G., DŽUBÁK P., ŠPENEROVÁ M., JANOŠŤÁKOVÁ A., FRYDRYCH I., KONEČNÝ P., OŽDIAN T., DOLEŽAL D., SOURAL M., HLAVÁČ J., HAJDÚCH M. Molecular targets and biological activity of quinolinone derivatives with anticancer effect. Optics Communications. 2011.
KONEČNÝ P., DŽUBÁK P., SOURAL M., HLAVÁČ J., FRYDRYCH I., RYLOVÁ G., KOCIS P., HAJDÚCH M. Profilování 2-fenylsubstituovaných-3-hydroxychinolin-4(1H)-one-karboxamidů a jejich protinádorových účinků metodou průtokové cytometrie. Optics Communications. 2011.
ŘEHULKA J., DŽUBÁK P., FRYDRYCH I., KREJČÍ P., SOURAL M., HAJDÚCH M. Selekce účinných 4-chinolonů s protinádorovou aktivitou a studium mechanizmu jejich účinku. Optics Communications. 2011.
Rylová G., Džubák P., Špenerová M., Janošťáková A., Frydrych I., Konečný P., Holub D., Oždian T., Doležal D., Soural M., Hlaváč J., Hajdúch M. Affinity purification coupled to mass spectrometry - approach to drug target identification. Onkologie - příloha Dny diagnostické, prediktivní a experimentální onkologie. 2010.
Frömmel J., Moskalíková H., Soural M., Tylichová M., Kopečný D., Šebela M. Exploring the active sites of plant aminoaldehyde dehydrogenases using natural and synthetic substrates. Sborník příspěvků (Book of Abstracts). 2010.
Frömmel J., Moskalíková H., Soural M., Tylichová M., Kopečný D., Šebela M. Exploring the active sites of plant aminoaldehyde dehydrogenases using natural and synthetic substrates. Materials Structure in Chemistry, Biology, Physics and Technology. 2010.
Rylová G., Džubák P., Špenerová M., Holub D., Oždian T., Soural M., Hlaváč J., Hajdúch M. Identifikace molekulárních cílů chinolonových derivátů pomocí afinitní purifikace spojené s LC-MSMS. Edukační sborník XXXIII. Brněnské onkologické dny. 2010.
Rylová G., Džubák P., Špenerová M., Holub D., Oždian T., Soural M., Hlaváč J., Hajdúch M. Molecular Targets Identification of Quinoline Derivatives by Affinity Purification Coupled to Mass Spectromentry. Sborník abstrakt - Biotechnologie v medicíně. 2010.
Rylová G., Džubák P., Špenerová M., Holub D., Oždian T., Soural M., Hlaváč J., Hajdúch M. Molecular targets identification of quinoline derivatives by affinity purification coupled to mass spectrometry. Book of Abstracts: Informal Proteomic Meeting 2010. 2010.
Frydrych I., Džubák P., Soural M., Hlaváč J., Funk P., Konečný P., Hajdúch M. 2-Substituted-3-Hydroxyquinoline-4(1H)-one-Carboxamides as potential anticancer drugs. Onkologie - příloha Dny diagnostické, prediktivní a experimentální onkologie. 2010.
Rylová G., Džubák P., Holub D., Špenerová M., Řehulka J., Soural M., Hlaváč J., Hajdúch M. AFFINITY PURIFICATION PROTEIN TARGETS OF ANTICANCER DRUGS AND THEIR. Sborník abstraktů přednášek MŠM 61989592. 2009.
Rylová G., Džubák P., Holub D., Špenerová M., Řehulka J., Soural M., Hlaváč J., Hajdúch M. Affinity purification protein targets of anticancer drugs and their identification by technology LC-MSMS. 3rd Central and Eastern European Proteomics Conference. Book of Abstracts and Program. 2009.
Rylová G., Džubák P., Holub D., Špenerová M., Soural M., Hlaváč J., Hajdúch M. Afinitní purifikace cílů protinádorových léčiv a jejich identifikace technologií LC-MALDI TOF-TOF. Konference vědeckých prací studentů DSP 2009. 2009.
Rylová G., Džubák P., Holub D., Špenerová M., Řehulka J., Soural M., Hlaváč J., Hajdúch M. New approach to target identification for anticancer drugs by LC-MSMS. Folia Medica Cassoviensia. 2009.
Klečková M., Pavlíček M., Štosová T., Cankař P., Soukupová J., Soural M., Vašíčková M. Tvorba korespondenčně - Internetové soutěže s chemickým zaměřením - Labyrint 2006. Nové metody propagace přírodních věd mezi mládeží (2006). 2006.
PŘEDNÁŠKA NEBO POSTER
Urban M., Borková L., Pokorný J., Džubák P., Hajdúch M., Soural M., Šarek J., Krajčovičová S., Řehulka J., Šidová V. Semisynthetic Triterpenes with Antitumor Activity – Synthesis, Cytotoxicity, and Studies of their Mechanism of Action. 2016.
KONFERENCE, WORKSHOP - USPOŘÁDÁNÍ
Štarha P., Drahoš B., Herchel R., Soural M., Plíhalová L., Bednář P., Panáček A. 12th Barrande-Vltava French-Czech Chemistry Meeting. 2023.

Uživatel nepovolil zobrazení dat v Portále UP.

Ph.D. studium na UP

Jméno Fakulta Studijní program Rok ukončení
FÜLÖPOVÁ PRF Chemie 2015
KRÁLOVÁ PRF Chemie 2020
LEMROVÁ PRF Chemie 2013
VANDA PRF Chemie 2021
KRAJČOVIČOVÁ PRF Chemie 2019
Seznam obsahuje absolventy úspěšně ukončeného doktorského studia.

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